Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50008268
TargetLysophosphatidic acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50517247(CHEMBL4442789)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human LPA1 expressed in CHO cells assessed as reduction in LPA-induced calcium influx incubated for 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50517246(CHEMBL4557434)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human LPA1 expressed in CHO cells assessed as reduction in LPA-induced calcium influx incubated for 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50517245(CHEMBL4442819)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at human LPA1 expressed in CHO cells assessed as reduction in LPA-induced calcium influx incubated for 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50517244(CHEMBL4448922)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human LPA1 expressed in CHO cells assessed as reduction in LPA-induced calcium influx incubated for 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50517248(CHEMBL4476814)
Affinity DataIC50: 227nMAssay Description:Antagonist activity at human LPA1 expressed in CHO cells assessed as reduction in LPA-induced calcium influx incubated for 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50517243(CHEMBL4472223)
Affinity DataIC50: 620nMAssay Description:Antagonist activity at human LPA1 expressed in CHO cells assessed as reduction in LPA-induced calcium influx incubated for 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed