Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50009157
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525822(CHEMBL4515933)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525814(CHEMBL4466132)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525810(CHEMBL4451680)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525815(CHEMBL4447048)
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525820(CHEMBL4457100)
Affinity DataIC50: 1.75E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525811(CHEMBL4474244)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525810(CHEMBL4451680)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525813(CHEMBL4579337)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525810(CHEMBL4451680)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525820(CHEMBL4457100)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525821(CHEMBL4526632)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525820(CHEMBL4457100)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525819(CHEMBL4538107)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525811(CHEMBL4474244)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525822(CHEMBL4515933)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525815(CHEMBL4447048)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525814(CHEMBL4466132)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525809(CHEMBL4552530)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525822(CHEMBL4515933)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525813(CHEMBL4579337)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525821(CHEMBL4526632)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525816(CHEMBL4533407)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525819(CHEMBL4538107)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525814(CHEMBL4466132)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525815(CHEMBL4447048)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525811(CHEMBL4474244)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525824(CHEMBL4527130)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525809(CHEMBL4552530)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525818(CHEMBL4592948)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525810(CHEMBL4451680)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]quinuclidinyl benzilate from Wistar rat cortex muscarinic acetylcholine receptor by liquid scintillation counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525827(CHEMBL4593317)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525817(CHEMBL4535766)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525826(CHEMBL4461203)
Affinity DataKi:  234nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525823(CHEMBL4467925)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525813(CHEMBL4579337)
Affinity DataKi:  454nMAssay Description:Displacement of [3H]quinuclidinyl benzilate from Wistar rat cortex muscarinic acetylcholine receptor by liquid scintillation counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525825(CHEMBL4520503)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525819(CHEMBL4538107)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]quinuclidinyl benzilate from Wistar rat cortex muscarinic acetylcholine receptor by liquid scintillation counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525812(CHEMBL4587692)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525821(CHEMBL4526632)
Affinity DataKi:  1.71E+3nMAssay Description:Displacement of [3H]quinuclidinyl benzilate from Wistar rat cortex muscarinic acetylcholine receptor by liquid scintillation counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50525820(CHEMBL4457100)
Affinity DataKi:  4.70E+3nMAssay Description:Displacement of [3H]quinuclidinyl benzilate from Wistar rat cortex muscarinic acetylcholine receptor by liquid scintillation counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed