Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50009434
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528834(CHEMBL4473727)
Affinity DataIC50: 37nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528838(CHEMBL4441237)
Affinity DataIC50: 41nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528835(CHEMBL4465796)
Affinity DataIC50: 50nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528841(CHEMBL4446234)
Affinity DataIC50: 55nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528822(CHEMBL4436169)
Affinity DataIC50: 55nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 55nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528825(CHEMBL4516296)
Affinity DataIC50: 57nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 59nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528840(CHEMBL4515881)
Affinity DataIC50: 62nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528836(CHEMBL4564320)
Affinity DataIC50: 71nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528819(CHEMBL4449161)
Affinity DataIC50: 79nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528821(CHEMBL4467130)
Affinity DataIC50: 80nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528831(CHEMBL4540497)
Affinity DataIC50: 84nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528832(CHEMBL4451686)
Affinity DataIC50: 94nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528824(CHEMBL4444516)
Affinity DataIC50: 102nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528833(CHEMBL4537886)
Affinity DataIC50: 114nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528828(CHEMBL4520782)
Affinity DataIC50: 135nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528823(CHEMBL4445907)
Affinity DataIC50: 148nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528829(CHEMBL4449791)
Affinity DataIC50: 151nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528826(CHEMBL4437163)
Affinity DataIC50: 172nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528830(CHEMBL4465315)
Affinity DataIC50: 174nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528839(CHEMBL4542575)
Affinity DataIC50: 216nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528827(CHEMBL4571434)
Affinity DataIC50: 226nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528820(CHEMBL4519129)
Affinity DataIC50: 276nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50528837(CHEMBL4519239)
Affinity DataIC50: 311nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed