Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50009151
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525789(CHEMBL4469854)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525789(CHEMBL4469854)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525793(CHEMBL4436129)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525793(CHEMBL4436129)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525797(CHEMBL4524344)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525797(CHEMBL4524344)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525795(CHEMBL4459383)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525795(CHEMBL4459383)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525790(CHEMBL4578823)
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525790(CHEMBL4578823)
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525796(CHEMBL4454551)
Affinity DataIC50: 102nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525796(CHEMBL4454551)
Affinity DataIC50: 103nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149992(CHEMBL3769897)
Affinity DataIC50: 157nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149992(CHEMBL3769897)
Affinity DataIC50: 158nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525792(CHEMBL4588969)
Affinity DataIC50: 162nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525792(CHEMBL4588969)
Affinity DataIC50: 162nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525794(CHEMBL4454980)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525794(CHEMBL4454980)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525791(CHEMBL4441341)
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50525791(CHEMBL4441341)
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human His-tagged GAC (72 to 603 residues) expressed in Escherichia coli using glutamine as substrate incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed