Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50008106
TargetPoly [ADP-ribose] polymerase 1(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of recombinant human full length N-terminal GST- tagged PARP1 expressed in baculovirus infected sf9 cells using Colorimetric HRP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPoly [ADP-ribose] polymerase 1(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50515712(CHEMBL4575720)
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant human full length N-terminal GST- tagged PARP1 expressed in baculovirus infected sf9 cells using Colorimetric HRP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50515710(CHEMBL4476017)
Affinity DataIC50: 350nMAssay Description:Inhibition of recombinant human full length N-terminal GST- tagged PARP1 expressed in baculovirus infected sf9 cells using Colorimetric HRP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50515715(CHEMBL4436472)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human full length N-terminal GST- tagged PARP1 expressed in baculovirus infected sf9 cells using Colorimetric HRP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50515711(CHEMBL4446682)
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of recombinant human full length N-terminal GST- tagged PARP1 expressed in baculovirus infected sf9 cells using Colorimetric HRP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50515713(CHEMBL4438977)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant human full length N-terminal GST- tagged PARP1 expressed in baculovirus infected sf9 cells using Colorimetric HRP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50515714(CHEMBL4563390)
Affinity DataIC50: 8.08E+3nMAssay Description:Inhibition of recombinant human full length N-terminal GST- tagged PARP1 expressed in baculovirus infected sf9 cells using Colorimetric HRP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed