Compile Data Set for Download or QSAR
Report error Found 138 Enz. Inhib. hit(s) with all data for entry = 50009606
Target5-hydroxytryptamine receptor 4(Human)
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Curated by ChEMBL
LigandPNGBDBM50530426(CHEMBL4557961)
Affinity DataEC50:  360nMAssay Description:Inhibition of 5-HT4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
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Curated by ChEMBL
LigandPNGBDBM50499430(CHEMBL3740472)
Affinity DataEC50:  22nMAssay Description:Inhibition of 5-HT4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
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Curated by ChEMBL
LigandPNGBDBM50530426(CHEMBL4557961)
Affinity DataEC50:  360nMAssay Description:Inhibition of 5-HT4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
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Curated by ChEMBL
LigandPNGBDBM50530443(CHEMBL4560185)
Affinity DataEC50:  72nMAssay Description:Inhibition of 5-HT4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
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Curated by ChEMBL
LigandPNGBDBM50530443(CHEMBL4560185)
Affinity DataEC50:  72nMAssay Description:Inhibition of 5-HT4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50499430(CHEMBL3740472)
Affinity DataEC50:  22nMAssay Description:Inhibition of 5-HT4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50397999(CHEMBL2180796)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50397999(CHEMBL2180796)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530441(CHEMBL4448109)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530441(CHEMBL4448109)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3(Human)
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Curated by ChEMBL
LigandPNGBDBM50386935(CHEMBL2048680)
Affinity DataIC50: 2nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3(Human)
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Curated by ChEMBL
LigandPNGBDBM50386935(CHEMBL2048680)
Affinity DataIC50: 2nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Human)
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Curated by ChEMBL
LigandPNGBDBM50530439(CHEMBL4456416)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Human)
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Curated by ChEMBL
LigandPNGBDBM50530439(CHEMBL4456416)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530425(CHEMBL4454665)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of FLAG-tagged human PDE4B2 expressed in Escherichia coli cells after 20 mins in presence of [3H]-cAMP by top count analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530425(CHEMBL4454665)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of FLAG-tagged human PDE4B2 expressed in Escherichia coli cells after 20 mins in presence of [3H]-cAMP by top count analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3(Human)
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Curated by ChEMBL
LigandPNGBDBM50386917(CHEMBL2048662)
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3(Human)
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Curated by ChEMBL
LigandPNGBDBM50530427(CHEMBL4562585)
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3(Human)
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Curated by ChEMBL
LigandPNGBDBM50386917(CHEMBL2048662)
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3(Human)
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Curated by ChEMBL
LigandPNGBDBM50530427(CHEMBL4562585)
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
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Curated by ChEMBL
LigandPNGBDBM269506((4-(2-chlorophenethyl)piperazin-1- yl)(imidazo[1,2...)
Affinity DataIC50: 4nMAssay Description:Modulator activity at 5-HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
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Curated by ChEMBL
LigandPNGBDBM269506((4-(2-chlorophenethyl)piperazin-1- yl)(imidazo[1,2...)
Affinity DataIC50: 4nMAssay Description:Modulator activity at 5-HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530417(CHEMBL4441878)
Affinity DataIC50: 6nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530417(CHEMBL4441878)
Affinity DataIC50: 6nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530430(CHEMBL4460561)
Affinity DataIC50: 7nMAssay Description:Inhibition of DYRK1A (unknown origin) by ADP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530430(CHEMBL4460561)
Affinity DataIC50: 7nMAssay Description:Inhibition of DYRK1A (unknown origin) by ADP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Human)
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Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Human)
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Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530429(CHEMBL4575900)
Affinity DataIC50: 8nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530429(CHEMBL4575900)
Affinity DataIC50: 8nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530417(CHEMBL4441878)
Affinity DataIC50: 9nMAssay Description:Inhibition of DYRK1A (unknown origin) by ADP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530417(CHEMBL4441878)
Affinity DataIC50: 9nMAssay Description:Inhibition of DYRK1A (unknown origin) by ADP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
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Curated by ChEMBL
LigandPNGBDBM50530423(CHEMBL4451349)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at 5-HT4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530423(CHEMBL4451349)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at 5-HT4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530430(CHEMBL4460561)
Affinity DataIC50: 11nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530430(CHEMBL4460561)
Affinity DataIC50: 11nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Human)
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Curated by ChEMBL
LigandPNGBDBM50060121(2-(6-Nitro-2-phenyl-imidazo[1,2-a]pyridin-3-yl)-N,...)
Affinity DataIC50: 12nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530429(CHEMBL4575900)
Affinity DataIC50: 12nMAssay Description:Inhibition of DYRK1A (unknown origin) by ADP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Human)
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Curated by ChEMBL
LigandPNGBDBM50060121(2-(6-Nitro-2-phenyl-imidazo[1,2-a]pyridin-3-yl)-N,...)
Affinity DataIC50: 12nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50530429(CHEMBL4575900)
Affinity DataIC50: 12nMAssay Description:Inhibition of DYRK1A (unknown origin) by ADP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3(Human)
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Curated by ChEMBL
LigandPNGBDBM50530444(CHEMBL4566900)
Affinity DataIC50: 13nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530444(CHEMBL4566900)
Affinity DataIC50: 13nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
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Curated by ChEMBL
LigandPNGBDBM50530422(CHEMBL4468363)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530422(CHEMBL4468363)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
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Curated by ChEMBL
LigandPNGBDBM50530429(CHEMBL4575900)
Affinity DataIC50: 19nMAssay Description:Inhibition of CLK1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
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Curated by ChEMBL
LigandPNGBDBM50530429(CHEMBL4575900)
Affinity DataIC50: 19nMAssay Description:Inhibition of CLK1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
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Curated by ChEMBL
LigandPNGBDBM50530417(CHEMBL4441878)
Affinity DataIC50: 20nMAssay Description:Inhibition of CLK1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530417(CHEMBL4441878)
Affinity DataIC50: 20nMAssay Description:Inhibition of CLK1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530430(CHEMBL4460561)
Affinity DataIC50: 21nMAssay Description:Inhibition of CLK1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530430(CHEMBL4460561)
Affinity DataIC50: 21nMAssay Description:Inhibition of CLK1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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