Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50008422
TargetSolute carrier family 15 member 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50519220(CHEMBL2229108)
Affinity DataIC50: 1.82E+7nMAssay Description:Substrate activity at PEPT1 in human Caco2 cells assessed as inhibition of Gly-Sar uptake measured after 10 mins by UPLC-MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50519221(CHEMBL4460144)
Affinity DataIC50: 1.76E+6nMAssay Description:Substrate activity at PEPT1 in human Caco2 cells assessed as inhibition of Gly-Sar uptake measured after 10 mins by UPLC-MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50519222(CHEMBL4540326)
Affinity DataIC50: 2.90E+6nMAssay Description:Substrate activity at PEPT1 in human Caco2 cells assessed as inhibition of Gly-Sar uptake measured after 10 mins by UPLC-MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50519221(CHEMBL4460144)
Affinity DataKi:  2.50E+6nMAssay Description:Substrate activity at PEPT1 in human Caco2 cells assessed as inhibition of Gly-Sar uptake by LC-MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50519220(CHEMBL2229108)
Affinity DataKi:  3.60E+7nMAssay Description:Substrate activity at PEPT1 in human Caco2 cells assessed as inhibition of Gly-Sar uptake by LC-MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed