Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50008764
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521959(CHEMBL4534481)
Affinity DataEC50: >3.57E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521965(CHEMBL4543257)
Affinity DataEC50:  460nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521964(CHEMBL4563335)
Affinity DataEC50:  1.39E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521963(CHEMBL4522441)
Affinity DataEC50:  1.24E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521962(CHEMBL4592654)
Affinity DataEC50:  1.45E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521961(CHEMBL4548269)
Affinity DataEC50:  2.41E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521960(CHEMBL4538761)
Affinity DataEC50: >4.01E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50085042(Finofibrate | Tricor (TN) | CHEMBL672 | propan-2-y...)
Affinity DataEC50:  5.00E+4nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521948(CHEMBL4454999)
Affinity DataEC50:  1.59E+4nMAssay Description:Transactivation of rat GAL4-fused PPARalpha expressed in human HepG2 cells after 24 hrs by dual renilla-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521948(CHEMBL4454999)
Affinity DataEC50:  1.13E+4nMAssay Description:Transactivation of mouse GAL4-fused PPARalpha expressed in human HepG2 cells after 24 hrs by dual renilla-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521948(CHEMBL4454999)
Affinity DataEC50:  660nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521958(CHEMBL4440299)
Affinity DataEC50:  1.53E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521957(CHEMBL4457812)
Affinity DataEC50:  680nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521956(CHEMBL4549332)
Affinity DataEC50:  1.80E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521955(CHEMBL4468865)
Affinity DataEC50:  2.06E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521954(CHEMBL4451764)
Affinity DataEC50:  1.98E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521953(CHEMBL4555785)
Affinity DataEC50:  1.23E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521952(CHEMBL4460143)
Affinity DataEC50: >1.34E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521951(CHEMBL4476019)
Affinity DataEC50: >2.27E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521950(CHEMBL4456624)
Affinity DataEC50: >2.74E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521949(CHEMBL4579518)
Affinity DataEC50:  1.76E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in human HepG2 cells after 24 hrs by renilla luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50521948(CHEMBL4454999)
Affinity DataIC50: 4.48E+3nMAssay Description:Displacement of fluormone pan-PPAR green from GST-tagged human PPARgamma ligand binding domain after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed