Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50007518
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50510090(CHEMBL4535730)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50510090(CHEMBL4535730)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50510091(CHEMBL4519542)
Affinity DataEC50:  1.69E+3nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50030474(US9562012, rosiglitazone | CHEBI:50122 | Avandamet...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50510092(CHEMBL4593987)
Affinity DataEC50:  184nMAssay Description:Agonist activity at human PPARalpha expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50510091(CHEMBL4519542)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50510093(CHEMBL4466552)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at human PPARalpha expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50510094(CHEMBL4460072)
Affinity DataEC50:  991nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50510092(CHEMBL4593987)
Affinity DataEC50:  84nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed