Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50008045
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515088(CHEMBL4447710)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515088(CHEMBL4447710)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK C481S mutant expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK C481S mutant expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515093(CHEMBL4541650)
Affinity DataIC50: 61nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK C481S mutant expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515091(CHEMBL4536906)
Affinity DataIC50: 73nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515093(CHEMBL4541650)
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515092(CHEMBL4552410)
Affinity DataIC50: 105nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515094(CHEMBL4543872)
Affinity DataIC50: 134nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515117(CHEMBL4455183)
Affinity DataIC50: 159nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515090(CHEMBL4584007)
Affinity DataIC50: 161nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515100(CHEMBL4454852)
Affinity DataIC50: 206nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515115(CHEMBL4472236)
Affinity DataIC50: 213nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515119(CHEMBL4450999)
Affinity DataIC50: 258nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515110(CHEMBL4587485)
Affinity DataIC50: 333nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515112(CHEMBL4564665)
Affinity DataIC50: 614nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515102(CHEMBL4579565)
Affinity DataIC50: 617nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515089(CHEMBL4460690)
Affinity DataIC50: 637nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515103(CHEMBL4548804)
Affinity DataIC50: 733nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515095(CHEMBL4460489)
Affinity DataIC50: 862nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515120(CHEMBL4528322)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515099(CHEMBL4562578)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515114(CHEMBL4441551)
Affinity DataIC50: 2.23E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515107(CHEMBL4450409)
Affinity DataIC50: 2.42E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515116(CHEMBL4547271)
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515111(CHEMBL4528929)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515118(CHEMBL4548153)
Affinity DataIC50: 5.17E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515113(CHEMBL4525695)
Affinity DataIC50: 5.25E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515105(CHEMBL4593580)
Affinity DataIC50: 5.32E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515101(CHEMBL4457726)
Affinity DataIC50: 6.75E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515096(CHEMBL4470618)
Affinity DataIC50: 8.53E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515098(CHEMBL4556566)
Affinity DataIC50: 1.92E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515106(CHEMBL4537375)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515087(CHEMBL4585613)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515108(CHEMBL4575423)
Affinity DataIC50: 2.78E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515109(CHEMBL4566033)
Affinity DataIC50: 3.71E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515104(CHEMBL4446069)
Affinity DataIC50: 3.81E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50515097(CHEMBL4476146)
Affinity DataIC50: 6.28E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His tagged BTK expressed in baculovirus infected Sf9 cells using poly (Glu,Tyr) 4:1 as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed