Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50008845
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataKd: 3.80E+3nMAssay Description:Binding affinity to N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in BL21 cells assessed as equilibrium dissociation constant ...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataKd: >5.00E+4nMAssay Description:Binding affinity to N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in BL21 cells assessed as equilibrium dissociation constant by ...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataKd: 720nMAssay Description:Binding affinity to N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in BL21 cells assessed as equilibrium dissociation constant ...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 4.76E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 4.37E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University
Curated by ChEMBL
Huazhong Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
