Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50005144
LigandPNGBDBM50502319(CHEMBL4515169)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50502315(CHEMBL4449091)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50502318(CHEMBL4542688)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50502321(CHEMBL4461362)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50502317(CHEMBL4471468)
Affinity DataIC50: 1nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50502320(CHEMBL4552869)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50502311(CHEMBL4439145)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PI3K delta (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50502324(CHEMBL4436369)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502316(CHEMBL4513335)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502325(CHEMBL4463308)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of PI3K delta (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50502315(CHEMBL4449091)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of PI3K gamma (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502311(CHEMBL4439145)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502315(CHEMBL4449091)
Affinity DataIC50: 5nMAssay Description:Inhibition of PI3K beta (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescenc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502323(CHEMBL4554487)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502318(CHEMBL4542688)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of PI3K beta (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescenc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502311(CHEMBL4439145)
Affinity DataIC50: 6nMAssay Description:Inhibition of PI3K gamma (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502318(CHEMBL4542688)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of PI3K gamma (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502315(CHEMBL4449091)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of PI3K delta (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502310(CHEMBL4470588)
Affinity DataIC50: 7nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502322(CHEMBL4227195)
Affinity DataIC50: 7nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502309(CHEMBL4441829)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502318(CHEMBL4542688)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of PI3K delta (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502312(CHEMBL4456355)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502326(CHEMBL4460217)
Affinity DataIC50: 12nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502311(CHEMBL4439145)
Affinity DataIC50: 16nMAssay Description:Inhibition of PI3K beta (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescenc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502313(CHEMBL4526257)
Affinity DataIC50: 34nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50502314(CHEMBL4460866)
Affinity DataIC50: 106nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50: 134nMAssay Description:Inhibition of PI3K beta (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescenc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM92862(mTOR Inhibitor, BEZ235 | US9284315, BEZ-235)
Affinity DataIC50: 169nMAssay Description:Inhibition of PI3K gamma (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM92862(mTOR Inhibitor, BEZ235 | US9284315, BEZ-235)
Affinity DataIC50: 204nMAssay Description:Inhibition of PI3K delta (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50: 381nMAssay Description:Inhibition of PI3K gamma (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM92862(mTOR Inhibitor, BEZ235 | US9284315, BEZ-235)
Affinity DataIC50: 421nMAssay Description:Inhibition of PI3K beta (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescenc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50: 583nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed