Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50010428
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538743(CHEMBL4640669)
Affinity DataKd:  1.28E+4nMAssay Description:Binding affinity to APC (unknown origin) by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538743(CHEMBL4640669)
Affinity DataIC50: 180nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538754(CHEMBL4641941)
Affinity DataIC50: 880nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538755(CHEMBL4635945)
Affinity DataIC50: 1.16E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538746(CHEMBL4644650)
Affinity DataIC50: 1.34E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538744(CHEMBL4647867)
Affinity DataIC50: 1.37E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538737(CHEMBL4637789)
Affinity DataIC50: 1.41E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538756(CHEMBL4647287)
Affinity DataIC50: 1.93E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538757(CHEMBL4647225)
Affinity DataIC50: 2.34E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538748(CHEMBL4632529)
Affinity DataIC50: 2.46E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538747(CHEMBL4642657)
Affinity DataIC50: 3.58E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538758(CHEMBL4632800)
Affinity DataIC50: 4.35E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538759(CHEMBL4646958)
Affinity DataIC50: 4.88E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538745(CHEMBL4646685)
Affinity DataIC50: 5.74E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538741(CHEMBL4643182)
Affinity DataIC50: 7.27E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538760(CHEMBL4633176)
Affinity DataIC50: 7.80E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538738(CHEMBL4646262)
Affinity DataIC50: 8.75E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538749(CHEMBL4649150)
Affinity DataIC50: 9.01E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538742(CHEMBL4647408)
Affinity DataIC50: 9.06E+3nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538752(CHEMBL4641939)
Affinity DataIC50: 1.40E+4nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538739(CHEMBL4638955)
Affinity DataIC50: 1.45E+4nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538761(CHEMBL4646420)
Affinity DataIC50: 1.56E+4nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538750(CHEMBL4645013)
Affinity DataIC50: 1.76E+4nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538753(CHEMBL4640305)
Affinity DataIC50: 1.99E+4nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538751(CHEMBL4641958)
Affinity DataIC50: 2.19E+4nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAdenomatous polyposis coli protein(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50538740(CHEMBL4649571)
Affinity DataIC50: 2.27E+4nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition of APC-Asef protein-protein interaction after 2 hrs by fluorescence polarization immu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed