Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50004438
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501984(CHEMBL4578651)
Affinity DataIC50: 4.30nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501982(CHEMBL4533857)
Affinity DataIC50: 4.30nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501969(CHEMBL4440692)
Affinity DataIC50: 4.70nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501986(CHEMBL4543370)
Affinity DataIC50: 5.30nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501980(CHEMBL4467767)
Affinity DataIC50: 5.30nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501971(CHEMBL4514580)
Affinity DataIC50: 5.70nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501985(CHEMBL4445475)
Affinity DataIC50: 5.70nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501973(CHEMBL4444248)
Affinity DataIC50: 6nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501975(CHEMBL4456486)
Affinity DataIC50: 6.30nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501979(CHEMBL4521251)
Affinity DataIC50: 7nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501974(CHEMBL4461157)
Affinity DataIC50: 7.30nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501978(CHEMBL4532018)
Affinity DataIC50: 7.70nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501981(CHEMBL4218019)
Affinity DataIC50: 8nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501983(CHEMBL4538025)
Affinity DataIC50: 9.30nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501970(CHEMBL4461263)
Affinity DataIC50: 11nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501977(CHEMBL4469374)
Affinity DataIC50: 12nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501976(CHEMBL4570799)
Affinity DataIC50: 13nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50501972(CHEMBL4443118)
Affinity DataIC50: 20nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50336730(4-[4-(2,4-Dioxothiazolidin-5-ylidenemethyl)-2-meth...)
Affinity DataIC50: 33nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50155833(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 61nMAssay Description:Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjugated coactivator PGC-1alpha incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50155833(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 370nMAssay Description:Inverse agonist activity at CMX-gal4-fused ERRgamma (unknown origin) transfected in (African Green monkey CV1 cells incubated for 20 hrs by luciferas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed