Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50008933
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50229962(N-(4-METHOXYBENZYL)-N'-(5-NITRO-1,3-THIAZOL-2-YL)U...)
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523726(CHEMBL4447545)
Affinity DataIC50: 86nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50229962(N-(4-METHOXYBENZYL)-N'-(5-NITRO-1,3-THIAZOL-2-YL)U...)
Affinity DataIC50: 104nMAssay Description:Inhibition of recombinant human GSK3alpha/beta using biotin-AAEELDSRAGS(PO3H2)PQL as substrate preincubated for 10 to 15 mins followed by [gamma-33P]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523722(CHEMBL1824333)
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523719(CHEMBL4546384)
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523724(CHEMBL4452731)
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523727(CHEMBL4532931)
Affinity DataIC50: 770nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523723(CHEMBL4516941)
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523725(CHEMBL4452831)
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523718(CHEMBL4556827)
Affinity DataIC50: 2.47E+3nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523721(CHEMBL4573681)
Affinity DataIC50: 4.05E+3nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523716(CHEMBL4571262)
Affinity DataIC50: 4.21E+3nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523717(CHEMBL4437756)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50523720(CHEMBL4461606)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using prephosphorylated peptide as substrate measured after 30 mins by Kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed