Compile Data Set for Download or QSAR
Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 50009068
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525095(CHEMBL4435895)
Affinity DataEC50:  794nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525097(CHEMBL4593181)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525097(CHEMBL4593181)
Affinity DataEC50:  7.94E+3nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM25771(salmeterol xinafoate | 4-(1-hydroxy-2-{[6-(4-pheny...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50167064(CHEMBL3797876)
Affinity DataEC50:  51nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50166977(CHEMBL3800303)
Affinity DataEC50:  501nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525095(CHEMBL4435895)
Affinity DataEC50:  398nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50407517(CHEMBL1160723 | (-)ISOPROTERENOL | US9492405, 27)
Affinity DataEC50:  50nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  251nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50166977(CHEMBL3800303)
Affinity DataEC50:  794nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525097(CHEMBL4593181)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50166977(CHEMBL3800303)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50167064(CHEMBL3797876)
Affinity DataEC50:  100nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50166977(CHEMBL3800303)
Affinity DataEC50:  100nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM25771(salmeterol xinafoate | 4-(1-hydroxy-2-{[6-(4-pheny...)
Affinity DataEC50:  0.0794nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  631nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50407517(CHEMBL1160723 | (-)ISOPROTERENOL | US9492405, 27)
Affinity DataEC50:  46nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50167064(CHEMBL3797876)
Affinity DataEC50:  158nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  794nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50407517(CHEMBL1160723 | (-)ISOPROTERENOL | US9492405, 27)
Affinity DataEC50:  25nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50407517(CHEMBL1160723 | (-)ISOPROTERENOL | US9492405, 27)
Affinity DataEC50:  20nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM25771(salmeterol xinafoate | 4-(1-hydroxy-2-{[6-(4-pheny...)
Affinity DataEC50:  0.126nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50407517(CHEMBL1160723 | (-)ISOPROTERENOL | US9492405, 27)
Affinity DataEC50:  44nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50167064(CHEMBL3797876)
Affinity DataEC50:  63nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  631nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50167064(CHEMBL3797876)
Affinity DataEC50:  63nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525095(CHEMBL4435895)
Affinity DataEC50:  794nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525097(CHEMBL4593181)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  316nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50167064(CHEMBL3797876)
Affinity DataEC50:  40nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525095(CHEMBL4435895)
Affinity DataEC50:  631nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525095(CHEMBL4435895)
Affinity DataEC50:  794nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50166977(CHEMBL3800303)
Affinity DataEC50:  794nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525095(CHEMBL4435895)
Affinity DataEC50:  316nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525097(CHEMBL4593181)
Affinity DataEC50:  1.26E+4nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525095(CHEMBL4435895)
Affinity DataEC50:  1.26E+4nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM25771(salmeterol xinafoate | 4-(1-hydroxy-2-{[6-(4-pheny...)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50407517(CHEMBL1160723 | (-)ISOPROTERENOL | US9492405, 27)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50407517(CHEMBL1160723 | (-)ISOPROTERENOL | US9492405, 27)
Affinity DataEC50:  25nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50167064(CHEMBL3797876)
Affinity DataEC50:  79nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50167064(CHEMBL3797876)
Affinity DataEC50:  269nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  316nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50407517(CHEMBL1160723 | (-)ISOPROTERENOL | US9492405, 27)
Affinity DataEC50:  52nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50166977(CHEMBL3800303)
Affinity DataEC50:  501nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50166977(CHEMBL3800303)
Affinity DataEC50:  417nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50166977(CHEMBL3800303)
Affinity DataEC50:  724nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525097(CHEMBL4593181)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM25771(salmeterol xinafoate | 4-(1-hydroxy-2-{[6-(4-pheny...)
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525095(CHEMBL4435895)
Affinity DataEC50:  398nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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