Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50010131
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50401993(CHEMBL2204696)
Affinity DataEC50:  6.40E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535438(CHEMBL4471853)
Affinity DataEC50:  380nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535435(CHEMBL4453610)
Affinity DataEC50:  3.90E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50401993(CHEMBL2204696)
Affinity DataEC50:  2.10E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535436(CHEMBL4449760)
Affinity DataEC50:  250nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535431(CHEMBL4557173)
Affinity DataEC50:  2.80E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50030474(US9562012, rosiglitazone | CHEBI:50122 | Avandamet...)
Affinity DataEC50:  40nMAssay Description:Transactivation of GAL4-tagged human PPARgamma LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535441(CHEMBL4461490)
Affinity DataEC50:  6.50E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535433(CHEMBL4461949)
Affinity DataEC50:  1.20E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535441(CHEMBL4461490)
Affinity DataEC50:  2.60E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535440(CHEMBL4438226)
Affinity DataEC50:  2.20E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50085041({4-[3-(4-acetyl-3-hydroxy-2-propylphenoxy)propoxy]...)
Affinity DataEC50:  210nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535439(CHEMBL4444322)
Affinity DataEC50:  2.30E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535436(CHEMBL4449760)
Affinity DataEC50:  6.00E+3nMAssay Description:Transactivation of GAL4-tagged human PPARgamma LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535430(CHEMBL4592451)
Affinity DataEC50:  2.40E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535438(CHEMBL4471853)
Affinity DataEC50:  3.10E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535434(CHEMBL4445737)
Affinity DataEC50:  1.80E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535437(CHEMBL4580572)
Affinity DataEC50:  4.10E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535436(CHEMBL4449760)
Affinity DataEC50:  2.80E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535432(CHEMBL4533822)
Affinity DataEC50:  1.10E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535435(CHEMBL4453610)
Affinity DataEC50:  810nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535434(CHEMBL4445737)
Affinity DataEC50:  2.30E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535433(CHEMBL4461949)
Affinity DataEC50:  510nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535432(CHEMBL4533822)
Affinity DataEC50:  1.90E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535431(CHEMBL4557173)
Affinity DataEC50:  1.40E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM28699(2-(4-chlorophenoxy)-2-methylpropanoic acid | CHEMB...)
Affinity DataEC50:  5.00E+4nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50535430(CHEMBL4592451)
Affinity DataEC50:  1.40E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed