Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50007282
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508113(CHEMBL4453360)
Affinity DataEC50:  2.72E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508124(CHEMBL4443588)
Affinity DataEC50:  1.53E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508112(CHEMBL4546437)
Affinity DataEC50:  1.73E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508123(CHEMBL4452865)
Affinity DataEC50:  3.31E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508122(CHEMBL4456647)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508121(CHEMBL4527893)
Affinity DataEC50:  2.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508120(CHEMBL4531918)
Affinity DataEC50:  2.62E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508119(CHEMBL4472191)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508118(CHEMBL4436393)
Affinity DataEC50:  7.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508117(CHEMBL4463602)
Affinity DataEC50:  2.53E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508116(CHEMBL4535401)
Affinity DataEC50:  2.78E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508115(CHEMBL4469751)
Affinity DataEC50:  1.81E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508114(CHEMBL4466241)
Affinity DataEC50:  1.32E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508101(CHEMBL4521388)
Affinity DataEC50:  1.66E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508111(CHEMBL4520827)
Affinity DataEC50:  460nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508110(CHEMBL4444760)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508109(CHEMBL4592935)
Affinity DataEC50:  1.03E+4nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508108(CHEMBL4567211)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508107(CHEMBL4574542)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508106(CHEMBL4517263)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508105(CHEMBL4542891)
Affinity DataEC50:  730nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508104(CHEMBL4591405)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508103(CHEMBL4589453)
Affinity DataEC50:  2.25E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508102(CHEMBL4537335)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508111(CHEMBL4520827)
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508110(CHEMBL4444760)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508112(CHEMBL4546437)
Affinity DataIC50: 440nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508112(CHEMBL4546437)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of human ERG by automated patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508112(CHEMBL4546437)
Affinity DataIC50: 7.50E+4nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508112(CHEMBL4546437)
Affinity DataIC50: 8.00E+4nMAssay Description:Binding affinity to PPARalpha (unknown origin) by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed