Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50003057
Target3-hydroxyacyl-CoA dehydrogenase type-2(Mouse)
Laval University

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 1.55E+5nMAssay Description:Inhibition of recombinant mouse full-length 17beta-HSD10 (2 to 261 residues) assessed as reduction in transformation of [14C]-E2 to E1 after 48 hrs i...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-hydroxyacyl-CoA dehydrogenase type-2(Mouse)
Laval University

Curated by ChEMBL
LigandPNGBDBM50466363(CHEMBL4277154)
Affinity DataIC50: 2.35E+5nMAssay Description:Inhibition of recombinant mouse full-length 17beta-HSD10 (2 to 261 residues) assessed as reduction in transformation of [3H]-ALLOP to 5alpha-DHP afte...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-hydroxyacyl-CoA dehydrogenase type-2(Mouse)
Laval University

Curated by ChEMBL
LigandPNGBDBM50466363(CHEMBL4277154)
Affinity DataIC50: 6.10E+5nMAssay Description:Inhibition of recombinant mouse full-length 17beta-HSD10 (2 to 261 residues) assessed as reduction in transformation of [14C]-E2 to E1 after 48 hrs i...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-hydroxyacyl-CoA dehydrogenase type-2(Mouse)
Laval University

Curated by ChEMBL
LigandPNGBDBM50466362(CHEMBL1813703)
Affinity DataIC50: 7.10E+5nMAssay Description:Inhibition of recombinant mouse full-length 17beta-HSD10 (2 to 261 residues) assessed as reduction in transformation of [14C]-E2 to E1 after 48 hrs i...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-hydroxyacyl-CoA dehydrogenase type-2(Mouse)
Laval University

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 7.70E+5nMAssay Description:Inhibition of recombinant mouse full-length 17beta-HSD10 (2 to 261 residues) assessed as reduction in transformation of [3H]-ALLOP to 5alpha-DHP afte...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-hydroxyacyl-CoA dehydrogenase type-2(Mouse)
Laval University

Curated by ChEMBL
LigandPNGBDBM50466362(CHEMBL1813703)
Affinity DataIC50: 9.85E+5nMAssay Description:Inhibition of recombinant mouse full-length 17beta-HSD10 (2 to 261 residues) assessed as reduction in transformation of [3H]-ALLOP to 5alpha-DHP afte...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed