Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50002509
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50403054(CHEMBL2216825)
Affinity DataIC50: 11nMAssay Description:Inhibition of ROCK2 (unknown origin) using SKT S2 as substrate measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50459504(CHEMBL4214797)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of ROCK2 (unknown origin) using SKT S2 as substrate measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50459501(CHEMBL4214283)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ROCK2 (unknown origin) using SKT S2 as substrate measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50459502(CHEMBL4209877)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ROCK2 (unknown origin) using SKT S2 as substrate measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50459503(CHEMBL4202607)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ROCK2 (unknown origin) using SKT S2 as substrate measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed