Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50002814
TargetHLA class I histocompatibility antigen, A alpha chain(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM86731(UK 33,274 | CAS_74191-85-8 | Doxazosin)
Affinity DataKd:  1.57E+4nMAssay Description:Binding affinity to human biotinylated HLA-A2 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetHLA class I histocompatibility antigen, A alpha chain(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM4851(cid_151194 | PTK787 | CHEMBL101253 | N-(4-chloroph...)
Affinity DataKd:  2.12E+4nMAssay Description:Binding affinity to human biotinylated HLA-A2 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetHLA class I histocompatibility antigen, A alpha chain(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM19441(Evista | CHEMBL81 | Keoxifene | Raloxifene, 6 | RA...)
Affinity DataKd:  2.20E+4nMAssay Description:Binding affinity to human biotinylated HLA-A2 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetHLA class I histocompatibility antigen, A alpha chain(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50073444(2-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}[1,2...)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to human biotinylated HLA-A2 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetHLA class I histocompatibility antigen, A alpha chain(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to human biotinylated HLA-A2 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetHLA class I histocompatibility antigen, A alpha chain(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKd: <1.00E+4nMAssay Description:Binding affinity to human biotinylated HLA-A2 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetHLA class I histocompatibility antigen, A alpha chain(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM24226(cid_2247 | [3H]-ASTEMIZOLE | Hismanal | ASTEMIZOLE...)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to human biotinylated HLA-A2 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed