Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50019137
Affinity DataKd: 0.170nMAssay Description:Inhibition of human RORgammmat LBD expressed in Escherichia coli by ThermoFluro assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human RORgammat expressed in COS7 cells by luciferase assayMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human GAL4-fused RORgammat LBD transfected in Escherichia coli BL21(DE3) cell measured after 16 hrs by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of RORgammat (unknown origin) by binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human GAL4-fused RORgammat LBD transfected in Escherichia coli BL21(DE3) cell measured after 16 hrs by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human RORgamma by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human RORgammat expressed in COS7 cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human GAL4-fused RORgammat LBD transfected in Escherichia coli BL21(DE3) cell measured after 16 hrs by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Inhibition of RORgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human GAL4-fused RORgammat LBD transfected in Escherichia coli BL21(DE3) cell measured after 16 hrs by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Inhibition of RORgamma LBD (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of His-tagged human RORgammat LBD in presence of biotin-coactivator peptide SRC1 binding incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of biotinylated human RORgammat by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Inhibition of RORgammat (unknown origin) by cell based reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Inhibition of human GAL4-fused RORgammat LBD transfected in Escherichia coli BL21(DE3) cell measured after 16 hrs by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human RORgammmat LBD expressed in Escherichia coli by FRET co-activator peptide assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of human RORgammmat LBD expressed in HEK293T by one-hybrid reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of His-tagged human RORgammat LBD in presence of biotin-coactivator peptide SRC1 binding incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inverse agonist activity at His-tagged human RORgammat LBD assessed as inhibition of biotinylated RIP140 co-activator peptide binding incubated for 1...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human RORgamma by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human RORgamma by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inverse agonist activity at GAL4-RORgammat LBD (unknown origin) expressed in HEK293 cells measured after 18 to 24 hrs by nuclear receptor assayMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of transactivation of Gal4-tagged RORgamma (unknown origin) transfected in human HG5LN cells incubated for 18 hrs by luciferase reporter g...More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of RORgammat (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inverse agonist activity at GAL4-tagged RORgammat (unknown origin) expressed in HEK293 cells measured after 18 hrs by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human RORgammmat LBD expressed in HEK293T by two-hybrid reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of RORgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of RORgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human RORgamma by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human GAL4-fused RORgamma LBD transfected in HEK293T cell measured after 24 hrs by luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human RORgamma by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human RORgamma by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of RORgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of human GAL4-fused RORgamma LBD transfected in HEK293T cell measured after 24 hrs by luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Inhibition of RORgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Antagonist activity at RORgammat LBD (unknown origin) assessed as fluorescent polarization signal measured in presence of fluorescein-labeled LXR ago...More data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Inhibition of human RORgammat expressed in COS7 cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of GAL4-RORgammat LBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Inhibition of human GAL4-fused RORgamma LBD transfected in HEK293T cell measured after 24 hrs by luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 245nMAssay Description:Inhibition of RORgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of human GAL4-fused RORgamma transfected in HEK293 cells co-transfected with G6Pase by luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of RORgammat LBD (unknown origin) expressed in Sf21 cells assessed as fluorescence signal by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inverse agonist activity at human GAL4-RORgamma DBD expressed in HEK293 cells measured after 24 hrs by ligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human GAL4-fused RORgamma LBD transfected in HEK293T cell measured after 24 hrs by luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human GAL4-fused RORalpha LBD transfected in HEK293T cell measured after 24 hrs by luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inverse agonist activity at human GAL4-RORgamma DBD expressed in HEK293 cells measured after 24 hrs by ligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inverse agonist activity at GAL4-tagged RORgammat (unknown origin) expressed in HEK293 cells measured after 18 hrs by luciferase assayMore data for this Ligand-Target Pair
Affinity DataKi: <100nMAssay Description:Inhibition of RORgamma (unknown origin)More data for this Ligand-Target Pair
