Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50001852
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: 74nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: 98nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: 290nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: 740nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: 760nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Pig)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406887(CHEMBL4162709)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406888(CHEMBL4175950)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406889(CHEMBL4168098)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406890(CHEMBL4173649)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Pig)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406892(CHEMBL4159749)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406989(CHEMBL4162053)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50407008(CHEMBL4170051)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406878(CHEMBL4166150)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406884(CHEMBL4168687)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406880(CHEMBL4170384)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406881(CHEMBL4177174)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Pig)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406886(CHEMBL4169579)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Pig)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Pig)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed