Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50001230
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Human)
University of Auckland
Curated by ChEMBL
University of Auckland
Curated by ChEMBL
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of BAPTA-induced Orai1-medited store operated calcium entry in human MDA-MB-231 cells pretreated for 15 mins followed by BAPTA addition by...More data for this Ligand-Target Pair
