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Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50002352
TargetLeukotriene A-4 hydrolase(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457473(CHEMBL4209822)
Affinity DataIC50: 8nMAssay Description:Inhibition of full-length recombinant C-terminal FLAG-tagged human leukotriene A4 hydrolase expressed in baculovirus-infected insect cells using Arg-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457479(CHEMBL1159812)
Affinity DataIC50: 11nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457478(CHEMBL4208547)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50368599(CHEMBL1159809)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457471(CHEMBL1159811)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457468(CHEMBL4216928)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50368598(CHEMBL1159810)
Affinity DataIC50: 21nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457469(CHEMBL4213478)
Affinity DataIC50: 25nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50131276(N-(3-{4-[3-(7-Chloro-quinolin-4-ylamino)-propyl]-p...)
Affinity DataIC50: 28nMAssay Description:Inhibition of APN in porcine kidney using Leu-p-NA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457473(CHEMBL4209822)
Affinity DataIC50: 30nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase using LGG as substrate after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457470(CHEMBL4204214)
Affinity DataIC50: 40nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457466(CHEMBL4206158)
Affinity DataIC50: 100nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase using LGG as substrate after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457473(CHEMBL4209822)
Affinity DataIC50: 190nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457466(CHEMBL4206158)
Affinity DataIC50: 220nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50089194(CHEMBL308333 | N*4*-Hydroxy-N*1*-[1-(2-hydroxymeth...)
Affinity DataIC50: 400nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50131276(N-(3-{4-[3-(7-Chloro-quinolin-4-ylamino)-propyl]-p...)
Affinity DataIC50: 854nMAssay Description:Inhibition of Plasmodium falciparum malaria M1 alanyl aminopeptidase using Leu-p-NA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457462(CHEMBL4212730)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of APN in porcine kidney microsomes using L-leucine-p-nitroanilide as substrate preincubated for 30 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457487(CHEMBL4207954)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of APN in porcine kidney microsomes using L-leucine-p-nitroanilide as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457480(CHEMBL4206336)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of APN in porcine kidney microsomes using L-leucine-p-nitroanilide as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457488(CHEMBL4217158)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457472(CHEMBL4213272)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457483(CHEMBL4217681)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of APN in porcine kidney microsomes using L-leucine-p-nitroanilide as substrate preincubated for 30 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of APN in porcine kidney microsomes using L-leucine-p-nitroanilide as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457483(CHEMBL4217681)
Affinity DataIC50: 2.03E+5nMAssay Description:Inhibition of recombinant human MMP2 expressed in Escherichia coli preincubated for 30 mins followed by succinylated gelatin substrate addition measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457465(CHEMBL4204736)
Affinity DataKi:  0.600nMAssay Description:Inhibition of APN in porcine kidney using Ala-p-NA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457475(CHEMBL4216408)
Affinity DataKi:  1.5nMAssay Description:Inhibition of APN in porcine kidney using Ala-p-NA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457479(CHEMBL1159812)
Affinity DataKi:  8nMAssay Description:Inhibition of APN in human placenta using AlabetaNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457482(CHEMBL4217064)
Affinity DataKi:  13nMAssay Description:Inhibition of APA (unknown origin) using GlubetaNA as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457485(CHEMBL4205440)
Affinity DataKi:  19nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457467(CHEMBL4217873)
Affinity DataKi:  19nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457477(CHEMBL4210855)
Affinity DataKi:  20nMAssay Description:Inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase [435-519](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50022748(2-Amino-4-methyl-pentane-1-thiol | CHEMBL69349)
Affinity DataKi:  22nMAssay Description:Competitive inhibition of LAP in porcine kidney microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036969((S)-2-Amino-pentane-1,5-dithiol | CHEMBL101771)
Affinity DataKi:  32nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036827([4-(2-Amino-3-mercapto-propyl)-cyclohexyl]-acetic ...)
Affinity DataKi:  35nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  36nMAssay Description:Inhibition of APN in porcine kidney using L-leucine p-nitroanilide as substrate preincubated for 60 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036968((S)-5-Amino-6-mercapto-hexanoic acid hydroxyamide ...)
Affinity DataKi:  37nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457478(CHEMBL4208547)
Affinity DataKi:  50nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  67nMAssay Description:Inhibition of APA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457476(CHEMBL4215801)
Affinity DataKi:  80nMAssay Description:Inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50121710(PIQ-22 | 2-(2,6-Diethyl-phenyl)-4H-isoquinoline-1,...)
Affinity DataKi:  120nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036824((S)-4-Amino-5-mercapto-pentanoic acid | (S)-3-Carb...)
Affinity DataKi:  120nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457482(CHEMBL4217064)
Affinity DataKi:  120nMAssay Description:Inhibition of APN in porcine kidney using Ala-betaNA as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457465(CHEMBL4204736)
Affinity DataKi:  130nMAssay Description:Inhibition of APA (unknown origin) using GluNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50089194(CHEMBL308333 | N*4*-Hydroxy-N*1*-[1-(2-hydroxymeth...)
Affinity DataKi:  170nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036962((S)-5-Amino-6-mercapto-hexanoic acid | (S)-4-Carbo...)
Affinity DataKi:  330nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50170890(CHEMBL3806072)
Affinity DataKi:  870nMAssay Description:Inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457479(CHEMBL1159812)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of APB in rat testis using ArgbetaNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457484(CHEMBL4206485)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of pig APNMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457474(CHEMBL4203613)
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of human APNMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
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