Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50002952
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50465075(CHEMBL4289425)
Affinity DataEC50:  111nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as reduction in amyloid beta (1 to 42) production after 60 mins by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50465076(CHEMBL4290617)
Affinity DataEC50:  19nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as reduction in amyloid beta (1 to 42) production after 60 mins by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50465077(CHEMBL4282341)
Affinity DataEC50:  14nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as reduction in amyloid beta (1 to 42) production after 60 mins by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50465078(CHEMBL4293906)
Affinity DataEC50:  35nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as reduction in amyloid beta (1 to 42) production after 60 mins by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50465079(CHEMBL4290214)
Affinity DataEC50:  34nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as reduction in amyloid beta (1 to 42) production after 60 mins by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50465080(CHEMBL4278756)
Affinity DataEC50:  36nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as reduction in amyloid beta (1 to 42) production after 60 mins by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed