Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50002630
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50460744(CHEMBL4227381)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50460750(CHEMBL4227461)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460756(CHEMBL4225346)
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460753(CHEMBL4228571)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460749(CHEMBL4229081)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460758(CHEMBL4225061)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460745(CHEMBL4228563)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460757(CHEMBL4225718)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460743(CHEMBL4229019)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460748(CHEMBL4226448)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460755(CHEMBL4226800)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460746(CHEMBL4228715)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460754(CHEMBL4229265)
Affinity DataIC50: 8.10nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460752(CHEMBL4226776)
Affinity DataIC50: 14nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460751(CHEMBL4229214)
Affinity DataIC50: 17nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460747(CHEMBL4226119)
Affinity DataIC50: 19nMAssay Description:Inhibition of PI3K p110delta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460745(CHEMBL4228563)
Affinity DataIC50: 25nMAssay Description:Inhibition of PI3K p110alpha (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460744(CHEMBL4227381)
Affinity DataIC50: 26nMAssay Description:Inhibition of PI3K p110alpha (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460753(CHEMBL4228571)
Affinity DataIC50: 27nMAssay Description:Inhibition of PI3K p110alpha (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50: 120nMAssay Description:Inhibition of PI3K p110beta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50: 139nMAssay Description:Inhibition of PI3K p110gamma (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460744(CHEMBL4227381)
Affinity DataIC50: 174nMAssay Description:Inhibition of PI3K p110gamma (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460753(CHEMBL4228571)
Affinity DataIC50: 199nMAssay Description:Inhibition of PI3K p110gamma (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460745(CHEMBL4228563)
Affinity DataIC50: 220nMAssay Description:Inhibition of PI3K p110beta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460745(CHEMBL4228563)
Affinity DataIC50: 224nMAssay Description:Inhibition of PI3K p110gamma (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460744(CHEMBL4227381)
Affinity DataIC50: 264nMAssay Description:Inhibition of PI3K p110beta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50: 306nMAssay Description:Inhibition of PI3K p110alpha (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460753(CHEMBL4228571)
Affinity DataIC50: 585nMAssay Description:Inhibition of PI3K p110beta (unknown origin) using lipid substrate after 40 mins by kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed