Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50002729
TargetKelch-like ECH-associated protein 1(Human)
University of East Anglia

Curated by ChEMBL
LigandPNGBDBM50462206(CHEMBL4248736)
Affinity DataKi:  6.10nMAssay Description:Displacement of F-14 from Keap1 Kelch domain (unknown origin) expressed in Escherichia coli BL21 (DE3) after 15 mins by fluorescence polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University of East Anglia

Curated by ChEMBL
LigandPNGBDBM50462209(CHEMBL4247618)
Affinity DataKi:  48nMAssay Description:Displacement of F-14 from Keap1 Kelch domain (unknown origin) expressed in Escherichia coli BL21 (DE3) after 15 mins by fluorescence polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University of East Anglia

Curated by ChEMBL
LigandPNGBDBM50462212(CHEMBL4239409)
Affinity DataKi:  48nMAssay Description:Displacement of F-14 from Keap1 Kelch domain (unknown origin) expressed in Escherichia coli BL21 (DE3) after 15 mins by fluorescence polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University of East Anglia

Curated by ChEMBL
LigandPNGBDBM50462207(CHEMBL4238711)
Affinity DataKi:  62nMAssay Description:Displacement of F-14 from Keap1 Kelch domain (unknown origin) expressed in Escherichia coli BL21 (DE3) after 15 mins by fluorescence polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University of East Anglia

Curated by ChEMBL
LigandPNGBDBM50462211(CHEMBL4250785)
Affinity DataKi:  95nMAssay Description:Displacement of F-14 from Keap1 Kelch domain (unknown origin) expressed in Escherichia coli BL21 (DE3) after 15 mins by fluorescence polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University of East Anglia

Curated by ChEMBL
LigandPNGBDBM50462208(CHEMBL4243641)
Affinity DataKi:  275nMAssay Description:Displacement of F-14 from Keap1 Kelch domain (unknown origin) expressed in Escherichia coli BL21 (DE3) after 15 mins by fluorescence polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University of East Anglia

Curated by ChEMBL
LigandPNGBDBM50462210(CHEMBL4238271)
Affinity DataKi:  1.52E+5nMAssay Description:Displacement of F-14 from Keap1 Kelch domain (unknown origin) expressed in Escherichia coli BL21 (DE3) after 15 mins by fluorescence polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed