Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50002619
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50360601(CHEMBL1933349 | MK-0893)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50168081(CHEMBL3799802 | MK 0893)
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460577(CHEMBL4229115)
Affinity DataIC50: 60nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460576(CHEMBL4224961)
Affinity DataIC50: 70nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50360601(CHEMBL1933349 | MK-0893)
Affinity DataIC50: 80nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460568(CHEMBL4227964)
Affinity DataIC50: 80nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460590(CHEMBL4227364)
Affinity DataIC50: 90nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50168081(CHEMBL3799802 | MK 0893)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460582(CHEMBL4227372)
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460591(CHEMBL4227229)
Affinity DataIC50: 110nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460578(CHEMBL4226972)
Affinity DataIC50: 180nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460583(CHEMBL4228215)
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460590(CHEMBL4227364)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460585(CHEMBL4227667)
Affinity DataIC50: 230nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460577(CHEMBL4229115)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460586(CHEMBL4227099)
Affinity DataIC50: 280nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460587(CHEMBL4228281)
Affinity DataIC50: 300nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460581(CHEMBL4227634)
Affinity DataIC50: 310nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460591(CHEMBL4227229)
Affinity DataIC50: 330nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460578(CHEMBL4226972)
Affinity DataIC50: 370nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460574(CHEMBL4225922)
Affinity DataIC50: 370nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460588(CHEMBL4228470)
Affinity DataIC50: 390nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460576(CHEMBL4224961)
Affinity DataIC50: 440nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460582(CHEMBL4227372)
Affinity DataIC50: 450nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460574(CHEMBL4225922)
Affinity DataIC50: 450nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460568(CHEMBL4227964)
Affinity DataIC50: 460nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460580(CHEMBL4226911)
Affinity DataIC50: 500nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460571(CHEMBL4227906)
Affinity DataIC50: 550nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460579(CHEMBL4226770)
Affinity DataIC50: 570nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460575(CHEMBL4228690)
Affinity DataIC50: 630nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460570(CHEMBL4225050)
Affinity DataIC50: 740nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460583(CHEMBL4228215)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460588(CHEMBL4228470)
Affinity DataIC50: 830nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460571(CHEMBL4227906)
Affinity DataIC50: 880nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460575(CHEMBL4228690)
Affinity DataIC50: 1.19E+3nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460587(CHEMBL4228281)
Affinity DataIC50: 1.29E+3nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460581(CHEMBL4227634)
Affinity DataIC50: 1.49E+3nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460585(CHEMBL4227667)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460573(CHEMBL4228703)
Affinity DataIC50: 1.92E+3nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460580(CHEMBL4226911)
Affinity DataIC50: 2.03E+3nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460586(CHEMBL4227099)
Affinity DataIC50: 2.31E+3nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460584(CHEMBL4227967)
Affinity DataIC50: 2.38E+3nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460573(CHEMBL4228703)
Affinity DataIC50: 2.69E+3nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460570(CHEMBL4225050)
Affinity DataIC50: 2.75E+3nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460584(CHEMBL4227967)
Affinity DataIC50: 2.79E+3nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460589(CHEMBL4227111)
Affinity DataIC50: 3.23E+3nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460569(CHEMBL4228938)
Affinity DataIC50: 3.90E+3nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460572(CHEMBL4227068)
Affinity DataIC50: 4.92E+3nMAssay Description:Displacement of [125I]-glucagon from wild type human glucagon receptor expressed in CHOK1 cells after 3 hrs by micro beta scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460569(CHEMBL4228938)
Affinity DataIC50: 5.52E+3nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50460589(CHEMBL4227111)
Affinity DataIC50: 7.53E+3nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293T cells assessed as inhibition of glucagon-induced cAMP accumulation after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
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