Compile Data Set for Download or QSAR
Report error Found 124 Enz. Inhib. hit(s) with all data for entry = 50002937
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464962(CHEMBL4290574)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464962(CHEMBL4290574)
Affinity DataIC50: 10nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50: 52nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464968(CHEMBL4290977)
Affinity DataIC50: 113nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464965(CHEMBL4294116)
Affinity DataIC50: 125nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50: 150nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464968(CHEMBL4290977)
Affinity DataIC50: 170nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464965(CHEMBL4294116)
Affinity DataIC50: 200nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464959(CHEMBL4280336)
Affinity DataIC50: 260nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464959(CHEMBL4280336)
Affinity DataIC50: 350nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464978(CHEMBL4283793)
Affinity DataIC50: 360nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464978(CHEMBL4283793)
Affinity DataIC50: 420nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464963(CHEMBL4292640)
Affinity DataIC50: 520nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464966(CHEMBL4294367)
Affinity DataIC50: 572nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-9(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50: 590nMAssay Description:Inhibition of human 20S immunoproteasome beta-1 using Ac-PAL-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464963(CHEMBL4292640)
Affinity DataIC50: 820nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464966(CHEMBL4294367)
Affinity DataIC50: 880nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464961(CHEMBL4287879)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464973(CHEMBL4280071)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464973(CHEMBL4280071)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464958(CHEMBL4279971)
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464961(CHEMBL4287879)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464974(CHEMBL4282422)
Affinity DataIC50: 2.13E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464961(CHEMBL4287879)
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-1 using Z-LLE-betaNA as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464958(CHEMBL4279971)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-1 using Z-LLE-betaNA as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464974(CHEMBL4282422)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-1 using Z-LLE-betaNA as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464970(CHEMBL4281477)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464961(CHEMBL4287879)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464970(CHEMBL4281477)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-1 using Z-LLE-betaNA as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464958(CHEMBL4279971)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-9(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464961(CHEMBL4287879)
Affinity DataIC50: 2.77E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-1 using Ac-PAL-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464970(CHEMBL4281477)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464963(CHEMBL4292640)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464961(CHEMBL4287879)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-9(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464970(CHEMBL4281477)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-1 using Ac-PAL-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464963(CHEMBL4292640)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464967(CHEMBL4285574)
Affinity DataIC50: 3.93E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464982(CHEMBL4290109)
Affinity DataIC50: 3.96E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-9(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464958(CHEMBL4279971)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-1 using Ac-PAL-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464960(CHEMBL4278967)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-9(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464963(CHEMBL4292640)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-1 using Ac-PAL-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464960(CHEMBL4278967)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-1 using Z-LLE-betaNA as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-9(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464960(CHEMBL4278967)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-1 using Ac-PAL-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50: 4.85E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464980(CHEMBL4289358)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-1 using Z-LLE-betaNA as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464967(CHEMBL4285574)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464982(CHEMBL4290109)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464960(CHEMBL4278967)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-9(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464974(CHEMBL4282422)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-1 using Ac-PAL-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
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