Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50001554
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284911(CHEMBL4171806)
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human eEF2K expressed in Escherichia coli using biotinylated myelin basic protein as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284575(CHEMBL4173539)
Affinity DataIC50: 360nMAssay Description:Inhibition of recombinant rat GST-tagged eEF2K expressed in Escherichia coli BL21 (DE3) cells using yeast eEF2 as substrate preincubated for 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50375667(TX-1918 | CHEMBL437612)
Affinity DataIC50: 440nMAssay Description:Inhibition of eEF2K in human A431 cells using eEF2 as substrate preincubated for 30 mins followed by ATP/[gamma-32P]-ATP addition measured after 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50053584(CHEMBL1977874)
Affinity DataIC50: 510nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284772(CHEMBL4161771)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284552(CHEMBL4175822)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284884(CHEMBL4174332)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284553(CHEMBL4159191)
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284781(CHEMBL4172410)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284550(CHEMBL4170891)
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284551(CHEMBL4165316)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284581(CHEMBL4176687)
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284567(CHEMBL4162960)
Affinity DataIC50: 1.94E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284549(CHEMBL4166070)
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284564(CHEMBL4169445)
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284626(CHEMBL4162623)
Affinity DataIC50: 2.26E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284574(CHEMBL4170948)
Affinity DataIC50: 2.38E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284568(CHEMBL4166413)
Affinity DataIC50: 2.75E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284554(CHEMBL4173263)
Affinity DataIC50: 2.84E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284578(CHEMBL4166679)
Affinity DataIC50: 2.93E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284560(CHEMBL4173954)
Affinity DataIC50: 3.12E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284627(CHEMBL4169894)
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284563(CHEMBL4168628)
Affinity DataIC50: 3.34E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284559(CHEMBL4175523)
Affinity DataIC50: 3.37E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284576(CHEMBL4159867)
Affinity DataIC50: 3.51E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284571(CHEMBL4160807)
Affinity DataIC50: 3.67E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284580(CHEMBL4175396)
Affinity DataIC50: 3.78E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284556(CHEMBL4172533)
Affinity DataIC50: 3.85E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284566(CHEMBL4162577)
Affinity DataIC50: 4.44E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284555(CHEMBL4166213)
Affinity DataIC50: 4.45E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284562(CHEMBL4165208)
Affinity DataIC50: 4.45E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284585(CHEMBL4173320)
Affinity DataIC50: 4.79E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284570(CHEMBL4172081)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284548(CHEMBL4174994)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284910(CHEMBL4163235)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284561(CHEMBL4175938)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284791(CHEMBL4161520)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284565(CHEMBL4169836)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284569(CHEMBL4167655)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284767(CHEMBL4161570)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284765(CHEMBL4164776)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284742(CHEMBL4170518)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284577(CHEMBL4167115)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284572(CHEMBL4168729)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284583(CHEMBL4159250)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284582(CHEMBL4169490)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284557(CHEMBL4163026)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284573(CHEMBL4161882)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284579(CHEMBL4177312)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50284558(CHEMBL4160702)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed