Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50000179
TargetEphrin type-A receptor 2(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50246750(CHEMBL4071045)
Affinity DataKd:  81nMAssay Description:Binding affinity to recombinant human GST-tagged EphA2 cytoplasmic domain (560 to 976 residues) expressed in baculovirus expression system by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2019
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50246750(CHEMBL4071045)
Affinity DataKd:  3.62E+3nMAssay Description:Binding affinity to AKT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2019
Entry Details Article
PubMed
TargetNF-kappa-B inhibitor alpha(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50246750(CHEMBL4071045)
Affinity DataKd:  741nMAssay Description:Binding affinity to NFKBIA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2019
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50246758(CHEMBL4093682)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of EphA2 autophosphorylation at Ser897 in human C13 cells after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2019
Entry Details Article
PubMed