Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50002107
TargetEstrogen receptor beta(Human)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor (ER)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]tamoxifen from antiestrogen binding site (AEBS)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50020285(CHEMBL955 | 3'-Methoxy-4'Hydroxyclomiphene | 4-{2-...)
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]tamoxifen from antiestrogen binding site (AEBS)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50020286(CHEMBL292185 | 4-{1-Chloro-2-[4-(2-diethylamino-et...)
Affinity DataIC50: 32nMAssay Description:Displacement of [3H]tamoxifen from antiestrogen binding site (AEBS)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM50020285(CHEMBL955 | 3'-Methoxy-4'Hydroxyclomiphene | 4-{2-...)
Affinity DataIC50: 780nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor (ER)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM50020286(CHEMBL292185 | 4-{1-Chloro-2-[4-(2-diethylamino-et...)
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor (ER)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed