Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50000841
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 39nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261639(CHEMBL4076689)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261633(CHEMBL4079032)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261638(CHEMBL4073779)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261640(CHEMBL4096865)
Affinity DataIC50: 160nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261634(CHEMBL4097045)
Affinity DataIC50: 170nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261643(CHEMBL4071061)
Affinity DataIC50: 190nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261644(CHEMBL4072244)
Affinity DataIC50: 360nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261636(CHEMBL4065185)
Affinity DataIC50: 450nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 490nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261642(CHEMBL4073566)
Affinity DataIC50: 520nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261637(CHEMBL4092847)
Affinity DataIC50: 560nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261641(CHEMBL4074351)
Affinity DataIC50: 680nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261635(CHEMBL4091890)
Affinity DataIC50: 780nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261637(CHEMBL4092847)
Affinity DataIC50: 4.96E+3nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261641(CHEMBL4074351)
Affinity DataIC50: 5.78E+3nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261635(CHEMBL4091890)
Affinity DataIC50: 6.54E+3nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261644(CHEMBL4072244)
Affinity DataIC50: 7.68E+3nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261642(CHEMBL4073566)
Affinity DataIC50: 7.98E+3nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261636(CHEMBL4065185)
Affinity DataIC50: 8.41E+3nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261643(CHEMBL4071061)
Affinity DataIC50: 9.23E+3nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261640(CHEMBL4096865)
Affinity DataIC50: 9.54E+3nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261638(CHEMBL4073779)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261634(CHEMBL4097045)
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261639(CHEMBL4076689)
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50261633(CHEMBL4079032)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of ovine COX1 assessed as reduction in PGH2 formation by measuring PGF2alpha by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed