Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50002302
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456866(CHEMBL4205489)
Affinity DataEC50:  890nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456883(CHEMBL4203455)
Affinity DataEC50:  160nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456884(CHEMBL4207270)
Affinity DataEC50:  230nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456885(CHEMBL4212156)
Affinity DataEC50:  500nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456886(CHEMBL4207312)
Affinity DataEC50:  4.60E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456887(CHEMBL4208677)
Affinity DataEC50:  170nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456888(CHEMBL4204346)
Affinity DataEC50:  300nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456889(CHEMBL4205786)
Affinity DataEC50:  460nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456890(CHEMBL4204808)
Affinity DataEC50:  200nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456867(CHEMBL4214183)
Affinity DataEC50:  290nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456891(CHEMBL4211625)
Affinity DataEC50:  1.13E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456892(CHEMBL4213613)
Affinity DataEC50:  290nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456893(CHEMBL4212948)
Affinity DataEC50:  1.30E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456882(CHEMBL4207808)
Affinity DataEC50:  330nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456894(CHEMBL4208388)
Affinity DataEC50:  7.08E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456895(CHEMBL4217013)
Affinity DataEC50:  210nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456896(CHEMBL4206729)
Affinity DataEC50:  140nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456897(CHEMBL4206337)
Affinity DataEC50:  170nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456898(CHEMBL4215129)
Affinity DataEC50:  7.00E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456899(CHEMBL4207681)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456900(CHEMBL4215125)
Affinity DataEC50:  2.60E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456901(CHEMBL4209218)
Affinity DataEC50:  490nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50394684(CHEMBL2165615)
Affinity DataEC50:  1.09E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as assessed as reduction in Km for glucose in presence of 5 mM glucose by G6PDH coupled ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456883(CHEMBL4203455)
Affinity DataEC50:  50nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as assessed as reduction in Km for glucose in presence of 5 mM glucose by G6PDH coupled ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456902(CHEMBL4210790)
Affinity DataEC50:  2.22E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456903(CHEMBL4203863)
Affinity DataEC50:  210nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456870(CHEMBL4213321)
Affinity DataEC50:  5.42E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456859(CHEMBL4202493)
Affinity DataEC50:  900nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456860(CHEMBL4216606)
Affinity DataEC50:  690nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456861(CHEMBL4204989)
Affinity DataEC50:  100nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456862(CHEMBL4204287)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456863(CHEMBL4216383)
Affinity DataEC50:  870nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456864(CHEMBL4202919)
Affinity DataEC50:  200nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456865(CHEMBL4217491)
Affinity DataEC50:  6.08E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456866(CHEMBL4205489)
Affinity DataEC50:  30nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as assessed as reduction in Km for glucose in presence of 5 mM glucose by G6PDH coupled ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456867(CHEMBL4214183)
Affinity DataEC50:  150nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as assessed as reduction in Km for glucose in presence of 5 mM glucose by G6PDH coupled ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50394684(CHEMBL2165615)
Affinity DataEC50:  930nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456868(CHEMBL4217208)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456869(CHEMBL4217728)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456858(CHEMBL4212777)
Affinity DataEC50:  8.42E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456871(CHEMBL4205913)
Affinity DataEC50:  320nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456872(CHEMBL4212586)
Affinity DataEC50:  890nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456873(CHEMBL4212033)
Affinity DataEC50:  1.09E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456874(CHEMBL4216481)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456875(CHEMBL4209159)
Affinity DataEC50:  820nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456876(CHEMBL4211616)
Affinity DataEC50:  230nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456877(CHEMBL4206856)
Affinity DataEC50:  90nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456878(CHEMBL4211227)
Affinity DataEC50:  2.23E+3nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456879(CHEMBL4215660)
Affinity DataEC50:  180nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHexokinase-4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456880(CHEMBL4210704)
Affinity DataEC50:  550nMAssay Description:Activation of recombinant human liver glucokinase 2 assessed as reduction in NADH production in presence of 5 mM glucose by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
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