Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 4
TargetAlpha-1A adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81980(CAS_87051-46-5 | NSC_65652 | Butanserin)
Affinity DataKi:  1.86nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81981(NSC_71255 | CAS_82190-91-8 | Flufylline | Flufylli...)
Affinity DataKi:  4.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataKi:  5.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81978(NSC_159037 | CAS_159037 | R 56413)
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81979(Guanabenz | NSC_3517 | NSC_65636 | CAS_5051-62-7 |...)
Affinity DataKi:  28.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKi:  72.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81980(CAS_87051-46-5 | NSC_65652 | Butanserin)
Affinity DataKi:  75.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81981(NSC_71255 | CAS_82190-91-8 | Flufylline | Flufylli...)
Affinity DataKi:  120nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataKi:  191nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81979(Guanabenz | NSC_3517 | NSC_65636 | CAS_5051-62-7 |...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81978(NSC_159037 | CAS_159037 | R 56413)
Affinity DataKi:  257nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81978(NSC_159037 | CAS_159037 | R 56413)
Affinity DataKi:  282nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKi:  295nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81981(NSC_71255 | CAS_82190-91-8 | Flufylline | Flufylli...)
Affinity DataKi:  417nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataKi:  631nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81979(Guanabenz | NSC_3517 | NSC_65636 | CAS_5051-62-7 |...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2017
Entry Details Article
PubMed