Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50000602
TargetGTPase KRas(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)
Affinity DataKd:  11nMAssay Description:Binding affinity to human N-terminal His/AVi-tagged biotinylated GTPase KRas G12D mutant (1 to 169 residues) expressed in Escherichia coli BL21 (DE3)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2019
Entry Details Article
PubMed
TargetGTPase KRas(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)
Affinity DataKd:  35nMAssay Description:Binding affinity to human N-terminal His/AVi-tagged biotinylated GTPase KRas G12C mutant expressed in Escherichia coli BL21 (DE3) in presence of GDP ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2019
Entry Details Article
PubMed
TargetGTPase KRas(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)
Affinity DataKd:  200nMAssay Description:Binding affinity to human wild type N-terminal His/AVi-tagged biotinylated KRas expressed in Escherichia coli BL21 (DE3) in presence of GTP by SPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2019
Entry Details Article
PubMed
TargetGTPase KRas(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)
Affinity DataKd:  250nMAssay Description:Binding affinity to human N-terminal His/AVi-tagged biotinylated GTPase KRas G12C mutant expressed in Escherichia coli BL21 (DE3) in presence of GTP ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2019
Entry Details Article
PubMed
TargetGTPase KRas(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)
Affinity DataKd:  200nMAssay Description:Binding affinity to human wild type N-terminal His/AVi-tagged biotinylated KRas expressed in Escherichia coli BL21 (DE3) in presence of GTP by SPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2019
Entry Details Article
PubMed
TargetGTPase KRas(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)
Affinity DataKd:  58nMAssay Description:Binding affinity to human wild type N-terminal His/AVi-tagged biotinylated KRas expressed in Escherichia coli BL21 (DE3) in presence of GDP by SPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2019
Entry Details Article
PubMed