Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50001339
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50431176(CHEMBL2332556)
Affinity DataIC50: 210nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276759(CHEMBL4161111)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276767(CHEMBL4172844)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276766(CHEMBL4164939)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276764(CHEMBL4169620)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276765(CHEMBL4174508)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276763(CHEMBL158116)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276760(CHEMBL155629)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50213690(2-Biphenyl-4-yl-4-methyl-octahydro-benzo[1,4]oxazi...)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276758(CHEMBL4163846)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276761(CHEMBL4159384)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276762(CHEMBL4167297)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM23926(5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetSqualene synthase(Rat)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50276768(CHEMBL4168364)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SQS in rat microsomes using [3H]-FPP as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by sci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed