Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50002271
TargetHistone acetyltransferase p300(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50456444(CHEMBL3734823)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of p300 (unknown origin) using H3 peptide and acetyl-coA as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50456440(CHEMBL4217391)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of p300 (unknown origin) using H3 peptide and acetyl-coA as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50456441(CHEMBL4212972)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of p300 (unknown origin) using H3 peptide and acetyl-coA as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50456442(CHEMBL4217912)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of p300 (unknown origin) using H3 peptide and acetyl-coA as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50456443(CHEMBL4205687)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of p300 (unknown origin) using H3 peptide and acetyl-coA as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50456444(CHEMBL3734823)
Affinity DataKi:  400nMAssay Description:Inhibition of VMA intein chitin binding domain-fused p300 HAT domain (1287 to 1652 residues) (unknown origin) expressed in Escherichia coli BL21(RIL)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed