Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50000530
TargetCasein kinase II subunit alpha/beta(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252622(CHEMBL4070389)
Affinity DataKd:  310nMAssay Description:Binding affinity to CK2alpha/beta (unknown origin) expressed in Escherichia coli BL21(DE3) by ITCMore data for this Ligand-Target Pair
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PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252622(CHEMBL4070389)
Affinity DataKd:  320nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252608(CHEMBL4088836)
Affinity DataKd:  2.50E+5nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252609(CHEMBL4104331)
Affinity DataKd:  2.50E+5nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252621(CHEMBL4086439)
Affinity DataKd:  1.64E+3nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
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PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252627(CHEMBL4100054)
Affinity DataKd:  6.29E+5nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252628(CHEMBL4082041)
Affinity DataKd:  5.00E+5nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252629(CHEMBL4061844)
Affinity DataKd:  5.20E+5nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50226518(3-aminobenzoic acid | 3-Aminobenzoesaeure | m-Amin...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252630(CHEMBL1161012)
Affinity DataKd:  5.80E+4nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252632(CHEMBL4105345)
Affinity DataKd:  3.00E+5nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252633(CHEMBL4089903)
Affinity DataKd:  2.70E+5nMAssay Description:Binding affinity to CK2alpha (unknown origin) by ITCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252622(CHEMBL4070389)
Affinity DataIC50: 370nMAssay Description:Inhibition of CK2alpha (unknown origin) using RRRADDSDDDD as substrate after 40 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha/beta(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252622(CHEMBL4070389)
Affinity DataIC50: 670nMAssay Description:Inhibition of CK2alpha/beta (unknown origin) expressed in Escherichia coli BL21(DE3) using RRRADDSDDDD as substrate after 40 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed