Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50000973
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50266776(CHEMBL4066553)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human ERG expressed in CHOK1 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50266762(CHEMBL218974)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of human ERG expressed in CHOK1 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2020
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50266762(CHEMBL218974)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes assessed as decrease in formation of 6beta-hydroxytestosterone from testosterone after 10 mins by LC-M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50266763(CHEMBL4069220)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG expressed in CHOK1 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2020
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50266763(CHEMBL4069220)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CYP3A4 in human liver microsomes assessed as decrease in formation of 6beta-hydroxytestosterone from testosterone after 10 mins by LC-M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2020
Entry Details Article
PubMed