Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50001000
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267312(CHEMBL4105040)
Affinity DataIC50: 900nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267314(CHEMBL4076896)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267313(CHEMBL4080816)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267311(CHEMBL4070159)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267312(CHEMBL4105040)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of recombinant His/FLAG-tagged Leishmania infantum TryR dimerization assessed as dimer disruption after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267327(CHEMBL4096399)
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of recombinant His/FLAG-tagged Leishmania infantum TryR dimerization assessed as dimer disruption after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267314(CHEMBL4076896)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of recombinant His/FLAG-tagged Leishmania infantum TryR dimerization assessed as dimer disruption after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267311(CHEMBL4070159)
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of recombinant His/FLAG-tagged Leishmania infantum TryR dimerization assessed as dimer disruption after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267313(CHEMBL4080816)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of recombinant His/FLAG-tagged Leishmania infantum TryR dimerization assessed as dimer disruption after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267327(CHEMBL4096399)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267315(CHEMBL4066988)
Affinity DataIC50: 4.74E+4nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267322(CHEMBL4071202)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267323(CHEMBL4092024)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267324(CHEMBL4067449)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267325(CHEMBL4088684)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267326(CHEMBL4078357)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267321(CHEMBL4104638)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267316(CHEMBL4080414)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267310(CHEMBL4097340)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant Leishmania infantum TryR preincubated for 10 mins followed by T[S]2 substrate addition and measured after 1 hr in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267326(CHEMBL4078357)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant His/FLAG-tagged Leishmania infantum TryR dimerization assessed as dimer disruption after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267325(CHEMBL4088684)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant His/FLAG-tagged Leishmania infantum TryR dimerization assessed as dimer disruption after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Instituto De Qu£Mica M£Dica (Iqm-Csic)

Curated by ChEMBL
LigandPNGBDBM50267310(CHEMBL4097340)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant His/FLAG-tagged Leishmania infantum TryR dimerization assessed as dimer disruption after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed