Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50000999
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267307(CHEMBL4085842)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267306(CHEMBL4096021)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267291(CHEMBL4098967)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267296(CHEMBL4104658)
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267304(CHEMBL4099377)
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267294(CHEMBL4097141)
Affinity DataIC50: 64nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267302(CHEMBL4066569)
Affinity DataIC50: 192nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267293(CHEMBL4080008)
Affinity DataIC50: 202nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267303(CHEMBL4086559)
Affinity DataIC50: 223nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267292(CHEMBL4080934)
Affinity DataIC50: 251nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267305(CHEMBL4077973)
Affinity DataIC50: 543nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)
Affinity DataIC50: 570nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by lonWorks Quattro analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267301(CHEMBL4082763)
Affinity DataIC50: 636nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267308(CHEMBL4094086)
Affinity DataIC50: 685nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267309(CHEMBL4067014)
Affinity DataIC50: 715nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267300(CHEMBL4087243)
Affinity DataIC50: 839nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267290(CHEMBL4099445)
Affinity DataIC50: 877nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267299(CHEMBL4092788)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267298(CHEMBL4069277)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Nanjing Normal University

Curated by ChEMBL
LigandPNGBDBM50267296(CHEMBL4104658)
Affinity DataIC50: 8.46E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by lonWorks Quattro analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed