Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50000075
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240170(CHEMBL4064816)
Affinity DataIC50: 9.40nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50419410(CHEMBL1915252)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240166(CHEMBL4060959)
Affinity DataIC50: 71nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240164(CHEMBL4066926)
Affinity DataIC50: 89nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240151(CHEMBL4096952)
Affinity DataIC50: 97nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240160(CHEMBL4099299)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240149(CHEMBL4094186)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240162(CHEMBL4061415)
Affinity DataIC50: 150nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240157(CHEMBL4083777)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240154(CHEMBL4088199)
Affinity DataIC50: 190nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240139(CHEMBL4089560)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240167(CHEMBL4067374)
Affinity DataIC50: 290nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240152(CHEMBL4069759)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240143(CHEMBL4081686)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240141(CHEMBL4091957)
Affinity DataIC50: 360nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240158(CHEMBL4089147)
Affinity DataIC50: 410nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240159(CHEMBL4081279)
Affinity DataIC50: 410nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240144(CHEMBL4095087)
Affinity DataIC50: 450nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240147(CHEMBL4064961)
Affinity DataIC50: 540nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240168(CHEMBL4099699)
Affinity DataIC50: 600nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240161(CHEMBL4088628)
Affinity DataIC50: 840nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240142(CHEMBL4071137)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240146(CHEMBL4078569)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240150(CHEMBL4061088)
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240165(CHEMBL4091562)
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240169(CHEMBL4067673)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240140(CHEMBL4097281)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240156(CHEMBL4062041)
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240163(CHEMBL4089248)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240155(CHEMBL4070667)
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240148(CHEMBL4073554)
Affinity DataIC50: 2.60E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240145(CHEMBL4102847)
Affinity DataIC50: 9.60E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed