Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50000074
TargetDNA topoisomerase 2-alpha(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM22984(Adriamycin | (8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated kinetoplast DNA decatenation after 60 mins by ethidium bromide staining based agarose gel electroph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50240132(CHEMBL4090898)
Affinity DataIC50: 4.88E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated kinetoplast DNA decatenation after 60 mins by ethidium bromide staining based agarose gel electroph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50240135(CHEMBL4066762)
Affinity DataIC50: 5.44E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated kinetoplast DNA decatenation after 60 mins by ethidium bromide staining based agarose gel electroph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50240137(CHEMBL4062965)
Affinity DataIC50: 7.08E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated kinetoplast DNA decatenation after 60 mins by ethidium bromide staining based agarose gel electroph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50240136(CHEMBL4064044)
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated kinetoplast DNA decatenation after 60 mins by ethidium bromide staining based agarose gel electroph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50240138(CHEMBL4093358)
Affinity DataIC50: 2.91E+4nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated kinetoplast DNA decatenation after 60 mins by ethidium bromide staining based agarose gel electroph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50240134(CHEMBL4094285)
Affinity DataIC50: 5.29E+4nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated kinetoplast DNA decatenation after 60 mins by ethidium bromide staining based agarose gel electroph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50240133(CHEMBL4082118)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated kinetoplast DNA decatenation after 60 mins by ethidium bromide staining based agarose gel electroph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50031046(Indeno[1,2-c]cinnolin-11-one | CHEMBL127717)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated kinetoplast DNA decatenation after 60 mins by ethidium bromide staining based agarose gel electroph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed