Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50000744
TargetTyrosine-protein kinase BTK(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50260042(CHEMBL4064534)
Affinity DataIC50: 911nMAssay Description:Inhibition of recombinant full length His-tagged human BTK cytoplasmic domain expressed in baculovirus expression system by Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50260042(CHEMBL4064534)
Affinity DataIC50: 1.79E+3nMAssay Description:Inhibition of recombinant full length His-tagged human PIM1 expressed in baculovirus expression system by Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50260042(CHEMBL4064534)
Affinity DataIC50: 2.42E+3nMAssay Description:Inhibition of recombinant full length His-tagged human BMX cytoplasmic domain expressed in baculovirus expression system by Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50260042(CHEMBL4064534)
Affinity DataIC50: 5.02E+3nMAssay Description:Inhibition of GST-tagged human DDR1 catalytic domain (440 to 876 residues) expressed in baculovirus expression system by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50260042(CHEMBL4064534)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant full length GST-tagged human PIM2 expressed in baculovirus expression system by Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50260042(CHEMBL4064534)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-tagged human DDR2 cytoplasmic domain (427 to 855 residues) expressed in baculovirus expression system by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed