Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50049266
Affinity DataIC50: 3.20nMAssay Description:Inhibition of EGFR (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of EGFR (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of EGFR (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of EGFR (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of EGFR (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 145nMAssay Description:Inhibition of EGFR (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 156nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of EGFR (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Xuzhou Medical University
Curated by ChEMBL
Xuzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of RAF (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Human)
Xuzhou Medical University
Curated by ChEMBL
Xuzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of VEGFR2 (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.37E+4nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of c-MET (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of c-MET (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Human)
Xuzhou Medical University
Curated by ChEMBL
Xuzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of VEGFR2 (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of EGFR (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of EGFR (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Xuzhou Medical University
Curated by ChEMBL
Xuzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of RAF (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of EGFR (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B (unknown origin) measured after 40 mins by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
