Compile Data Set for Download or QSAR
Report error Found 91 Enz. Inhib. hit(s) with all data for entry = 50003214
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50015640(LY-2157299 | GALUNISERTIB)
Affinity DataIC50: 51nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468220(CHEMBL4277021)
Affinity DataIC50: 80nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468197(CHEMBL4285400)
Affinity DataIC50: 97nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468203(CHEMBL4287654)
Affinity DataIC50: 98nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468207(CHEMBL4288745)
Affinity DataIC50: 137nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468201(CHEMBL4292491)
Affinity DataIC50: 147nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468206(CHEMBL4291675)
Affinity DataIC50: 154nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468204(CHEMBL4289487)
Affinity DataIC50: 162nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50151347(2-(3-(6-methylpyridin-2-yl)-1H-pyrazol-4-yl)-1,5-n...)
Affinity DataIC50: 181nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468218(CHEMBL4279935)
Affinity DataIC50: 181nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468213(CHEMBL4281030)
Affinity DataIC50: 183nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468215(CHEMBL4277446)
Affinity DataIC50: 197nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468196(CHEMBL4291439)
Affinity DataIC50: 229nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468202(CHEMBL4279172)
Affinity DataIC50: 229nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468195(CHEMBL4283308)
Affinity DataIC50: 261nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468208(CHEMBL4278812)
Affinity DataIC50: 341nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468217(CHEMBL4276896)
Affinity DataIC50: 406nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468214(CHEMBL4284434)
Affinity DataIC50: 517nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468193(CHEMBL4287843)
Affinity DataIC50: 548nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468206(CHEMBL4291675)
Affinity DataIC50: 550nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468219(CHEMBL4292170)
Affinity DataIC50: 612nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468221(CHEMBL4292878)
Affinity DataIC50: 743nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468199(CHEMBL4284266)
Affinity DataIC50: 805nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468211(CHEMBL4284609)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468194(CHEMBL4287261)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468200(CHEMBL4282287)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468209(CHEMBL4285692)
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468210(CHEMBL4281195)
Affinity DataIC50: 1.99E+3nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468212(CHEMBL4294411)
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468201(CHEMBL4292491)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468205(CHEMBL4277755)
Affinity DataIC50: 2.52E+3nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468198(CHEMBL4287412)
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTGF-beta receptor type-1(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468216(CHEMBL4279331)
Affinity DataIC50: 5.19E+3nMAssay Description:Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468204(CHEMBL4289487)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468202(CHEMBL4279172)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50468206(CHEMBL4291675)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human CDK2/cyclin E expressed in Sf9 insect cells using histone H1 as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468194(CHEMBL4287261)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50468208(CHEMBL4278812)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human CDK2/cyclin E expressed in Sf9 insect cells using histone H1 as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468216(CHEMBL4279331)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468208(CHEMBL4278812)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50468216(CHEMBL4279331)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human CDK2/cyclin E expressed in Sf9 insect cells using histone H1 as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468196(CHEMBL4291439)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468205(CHEMBL4277755)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50151347(2-(3-(6-methylpyridin-2-yl)-1H-pyrazol-4-yl)-1,5-n...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468218(CHEMBL4279935)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468221(CHEMBL4292878)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468193(CHEMBL4287843)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50468215(CHEMBL4277446)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human CDK2/cyclin E expressed in Sf9 insect cells using histone H1 as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase ABL1(Mouse)
Palack£

Curated by ChEMBL
LigandPNGBDBM50468217(CHEMBL4276896)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of mouse ABL expressed in Sf9 insect cells using GGEAIYAAPFKK as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50468202(CHEMBL4279172)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of human CDK2/cyclin E expressed in Sf9 insect cells using histone H1 as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 91 total ) | Next | Last >>
Jump to: