Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50049190
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50385568(CHEMBL2040640)
Affinity DataIC50: 190nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) PA endonuclease using ALMV cap1 primer RNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50385503(CHEMBL2040554)
Affinity DataIC50: 320nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) PA endonuclease using ALMV cap1 primer RNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50122448(L-742001 | CHEMBL463590)
Affinity DataIC50: 430nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) PA endonuclease using ALMV cap1 primer RNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50385528(CHEMBL2040586)
Affinity DataIC50: 540nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) PA endonuclease using ALMV cap1 primer RNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50385531(CHEMBL2040602)
Affinity DataIC50: 800nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) N-terminal PA endonuclease using 880 nucleotide ALMV cap1 primer RNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50125833(3-(4-Fluoro-benzylidene)-1-hydroxy-5-isobutyl-3H-p...)
Affinity DataIC50: 900nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) N-terminal PA endonuclease using 880 nucleotide ALMV cap1 primer RNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50385529(CHEMBL2040587)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) PA endonuclease using ALMV cap1 primer RNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50385534(CHEMBL2040605)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) N-terminal PA endonuclease using 880 nucleotide ALMV cap1 primer RNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50385535(CHEMBL2040606)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) N-terminal PA endonuclease using 880 nucleotide ALMV cap1 primer RNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50125822(1-Hydroxy-5-isobutyl-3-isobutylidene-3H-pyrazine-2...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) N-terminal PA endonuclease using 880 nucleotide ALMV cap1 primer RNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Shandong University

Curated by ChEMBL
LigandPNGBDBM33410(CHEMBL16755 | N-hydroxyisoquinolinedione, 2)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of influenza A virus (A/PR/8/34) PA endonuclease using ALMV cap1 primer RNA as substrate after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)