Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50048938
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230303(CHEMBL3990703)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230310(CHEMBL4091587)
Affinity DataEC50:  1.14E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230309(CHEMBL4071849)
Affinity DataEC50:  1.11E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230308(CHEMBL4072869)
Affinity DataEC50:  1.27E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230307(CHEMBL4083311)
Affinity DataEC50:  2.56E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230306(CHEMBL4073421)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 2(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230295(CHEMBL4098843)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 3(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230295(CHEMBL4098843)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FFA3 receptor expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230304(CHEMBL4101306)
Affinity DataEC50:  6.10E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230295(CHEMBL4098843)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230302(CHEMBL4077784)
Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230301(CHEMBL4064196)
Affinity DataEC50:  3.35E+4nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230300(CHEMBL4101806)
Affinity DataEC50:  2.36E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230299(CHEMBL4063785)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230298(CHEMBL4063221)
Affinity DataEC50:  1.48E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230297(CHEMBL4091100)
Affinity DataEC50:  1.21E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230295(CHEMBL4098843)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50230296(CHEMBL4093571)
Affinity DataEC50:  3.87E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium flux by Fluo-8 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2019
Entry Details Article
PubMed